SCHEMBL8725587

SCHEMBL8725587

CC(OC(=O)CCCc1cccs1)[C@H]1CC[C@H]2[C@@H]3CCN4C(C)C(=O)CC[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.36
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
GPBAR1 Q8TDU6 2/20 0.33
PTPN1 P18031 1/20 0.33
CYP2C9 P11712 1/20 0.33
HIF1A Q16665 1/20 0.33
VDR P11473 1/20 0.33
EBP Q15125 1/20 0.32
DHCR7 Q9UBM7 1/20 0.32
SRD5A2 P31213 1/20 0.32
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8931575 0.82 FNTA (0.36) FNTAFNTBGPBAR1CYP2C9HIF1A
SCHEMBL7749997 0.81 SRD5A1 (0.52) SRD5A2
SCHEMBL7750005 0.81 SRD5A1 (0.52) SRD5A2
SCHEMBL9114171 0.81 FAAH (0.38) FNTAFNTBGPBAR1CYP2C9HIF1A
SCHEMBL8726712 0.80 ALDH1A1 (0.39) NR1H4SRD5A2
SCHEMBL8722384 0.80 FNTA (0.35) FNTAFNTBGPBAR1CYP2C9HIF1A
SCHEMBL9113840 0.77 GPBAR1 (0.36) FNTAFNTBGPBAR1SRD5A2
SCHEMBL9113437 0.76 SRD5A2 (0.36) FNTAFNTBGPBAR1SRD5A2
SCHEMBL9113792 0.75 GPBAR1 (0.36) GPBAR1CYP2C9HIF1AVDRSRD5A2
SCHEMBL7745521 0.75 RORC (0.36) FNTAFNTBGPBAR1CYP2C9HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710275-A ENZYME AND HORMONE INHIBITORS MERCK & CO., INC. (US) 1998-01-20 US disclosed
EP-0778284-A2 New 7-beta-substituted-4-aza-5alpha-androstan-3-ones as 5alpha-reductase inhibitors MERCK & CO. INC. (US) 1997-06-11 EP disclosed
EP-0572166-A1 New 7beta-substituted-4-aza-5a-androstan-3-ones as 5a-reductase inhibitors MERCK & CO. INC. (US) 1993-12-01 EP disclosed