SCHEMBL8727207

SCHEMBL8727207

[c]1ccccc1Nc1ccc(CCn2cnnn2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HMOX1 P09601 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
TP53 P04637 4/20 0.40
ALDH1A1 P00352 4/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
RAB9A P51151 1/20 0.36
MAPT P10636 2/20 0.34
MAPK1 P28482 2/20 0.34
LTA4H P09960 1/20 0.33
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
THRB P10828 1/20 0.33
GAA P10253 1/20 0.32
KDM4E B2RXH2 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
TNIK Q9UKE5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8727211 0.83 HRH3 (0.43) HMOX1HRH3TP53ALDH1A1MEN1
SCHEMBL8727126 0.72 CYP19A1 (0.55)
SCHEMBL8722545 0.71 SLC6A4 (0.49) LTA4H
SCHEMBL8723594 0.69 HRH3 (0.44) HRH3MAPK1LTA4HKDM4E
SCHEMBL8722523 0.69 TSHR (0.40) ALDH1A1MAPK1LTA4HL3MBTL1
SCHEMBL6880513 0.69 MEN1 (0.52) HMOX1HRH3TP53ALDH1A1MEN1
SCHEMBL6880509 0.69 ALDH1A1 (0.52) HMOX1HRH3TP53ALDH1A1MEN1
SCHEMBL29788842 0.69 RAB9A (0.52) HMOX1HRH3TP53ALDH1A1MEN1
SCHEMBL8722517 0.68 CYP11B1 (0.56) MAPTPOLB
SCHEMBL29788848 0.66 HMOX1 (0.56) HMOX1TP53ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed