SCHEMBL8729317

SCHEMBL8729317

CN(C(=O)NC(Cc1ccccc1)C(O)C(N)(Cc1ccccc1)C(=O)NC(C)(C)C)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
BCHE P06276 3/20 0.36
KLK5 Q9Y337 3/20 0.36
BACE1 P56817 5/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
RECQL P46063 1/20 0.35
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
CTSD P07339 1/20 0.35
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8734199 0.93 MMP1 (0.38) OPRM1OPRD1PSEN1PSEN2APH1B
SCHEMBL8729332 0.92 BCHE (0.36) OPRM1OPRD1OPRK1PSEN1PSEN2
SCHEMBL8734156 0.91 MME (0.40) CTSD
SCHEMBL8729353 0.90 MMP2 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8732148 0.90 PSEN1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8734166 0.88 BACE1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8882496 0.88 PSEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8734448 0.73 BCHE (0.65) BCHEBACE1CTSD
SCHEMBL8729411 0.72 BACE1 (0.61) BCHEBACE1CTSD
SCHEMBL8840094 0.71 PSEN1 (0.51) OPRM1OPRD1OPRK1PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708004-A ENZYME INHIBITORS FOR TREATMENT OF AIDS MONSANTO COMPANY (US) 1998-01-13 US disclosed
US-5703076-A TREATING HIV, AIDS G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
US-5698569-A Retroviral protease inhibitors G. D. SEARLE & CO. (US) 1997-12-16 US disclosed
US-5510349-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510378-A Retroviral protease inhibitors G.D. SEARLE & CO. (US) 1996-04-23 US disclosed