SCHEMBL8734156

SCHEMBL8734156

CN(C(=O)NC(Cc1ccccc1)C(O)C(N)(Cc1ccc2ccccc2c1)C(=O)NC(C)(C)C)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MME P08473 4/20 0.40
ACE P12821 3/20 0.40
CASR P41180 3/20 0.38
FCER2 P06734 4/20 0.37
MMP9 P14780 2/20 0.37
CTSD P07339 2/20 0.36
CCR1 P32246 1/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
CAPN1 P07384 1/20 0.35
MMP8 P22894 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729317 0.91 OPRM1 (0.38) CTSD
SCHEMBL8734199 0.88 MMP1 (0.38) MMP9
SCHEMBL8729332 0.85 BCHE (0.36) CTSD
SCHEMBL8734166 0.84 BACE1 (0.36) CTSD
SCHEMBL8732148 0.83 PSEN1 (0.37)
SCHEMBL8729353 0.83 MMP2 (0.37) CTSD
SCHEMBL8882496 0.82 PSEN1 (0.38) MMEACECTSD
SCHEMBL8731396 0.77 BACE1 (0.54) CTSD
SCHEMBL8840008 0.74 PSEN1 (0.45) MMEACECTSDCYP2D6SLC6A3
SCHEMBL6223038 0.74 PSEN1 (0.45) MMEACECTSDCYP2D6SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708004-A ENZYME INHIBITORS FOR TREATMENT OF AIDS MONSANTO COMPANY (US) 1998-01-13 US disclosed
US-5703076-A TREATING HIV, AIDS G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
US-5698569-A Retroviral protease inhibitors G. D. SEARLE & CO. (US) 1997-12-16 US disclosed
US-5510349-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510487-A TREATING HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510378-A Retroviral protease inhibitors G.D. SEARLE & CO. (US) 1996-04-23 US disclosed