SCHEMBL8734199

SCHEMBL8734199

COc1ccc(CC(N)(C(=O)NC(C)(C)C)C(O)C(Cc2ccccc2)NC(=O)N(C)c2ccccc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 6/20 0.38
MMP13 P45452 2/20 0.38
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38
MMP3 P08254 3/20 0.38
MMP9 P14780 3/20 0.38
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
ATM Q13315 1/20 0.36
CNR2 P34972 1/20 0.36
PSEN1 P49768 2/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
KMT2A Q03164 1/20 0.36
NPY5R Q15761 1/20 0.36
FPR2 P25090 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729317 0.93 OPRM1 (0.38) ITGA4ITGB7OPRM1OPRD1PSEN1
SCHEMBL8734156 0.88 MME (0.40) MMP9
SCHEMBL8729332 0.85 BCHE (0.36) ITGA4ITGB7MMP3OPRM1OPRD1
SCHEMBL8732148 0.83 PSEN1 (0.37) ITGA4ITGB7PSEN1PSEN2APH1B
SCHEMBL8729353 0.83 MMP2 (0.37) MMP1ITGA4ITGB7MMP3PSEN1
SCHEMBL8882496 0.82 PSEN1 (0.38) MMP3PSEN1PSEN2APH1BNCSTN
SCHEMBL8734166 0.82 BACE1 (0.36) ITGA4ITGB7MMP3CNR2PSEN1
SCHEMBL8734182 0.77 BCHE (0.56)
SCHEMBL3351385 0.69 BCHE (0.69)
SCHEMBL3351378 0.69 BCHE (0.69)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708004-A ENZYME INHIBITORS FOR TREATMENT OF AIDS MONSANTO COMPANY (US) 1998-01-13 US disclosed
US-5703076-A TREATING HIV, AIDS G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
US-5698569-A Retroviral protease inhibitors G. D. SEARLE & CO. (US) 1997-12-16 US disclosed
US-5510349-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510378-A Retroviral protease inhibitors G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510487-A TREATING HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed