SCHEMBL8732148

SCHEMBL8732148

CC(C)CC(N)(C(=O)NC(C)(C)C)C(O)C(Cc1ccccc1)NC(=O)N(C)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 9/20 0.37
PSEN2 P49810 9/20 0.37
APH1B Q8WW43 9/20 0.37
NCSTN Q92542 9/20 0.37
APH1A Q96BI3 9/20 0.37
PSENEN Q9NZ42 9/20 0.37
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
ACACB O00763 1/20 0.34
KLK5 Q9Y337 1/20 0.34
ITGA4 P13612 1/20 0.34
ITGB7 P26010 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PSMB1 P20618 1/20 0.33
PSMB5 P28074 1/20 0.33
PSMB2 P49721 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8882496 0.90 PSEN1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8729332 0.90 BCHE (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8729317 0.90 OPRM1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8729353 0.88 MMP2 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8734166 0.87 BACE1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8734156 0.83 MME (0.40)
SCHEMBL8734199 0.83 MMP1 (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL8729343 0.79 LAP3 (0.45) NPC1RAB9A
SCHEMBL8731465 0.71 BACE1 (0.50)
SCHEMBL7322817 0.71 BACE1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708004-A ENZYME INHIBITORS FOR TREATMENT OF AIDS MONSANTO COMPANY (US) 1998-01-13 US disclosed
US-5703076-A TREATING HIV, AIDS G. D. SEARLE & CO. (US) 1997-12-30 US disclosed
US-5698569-A Retroviral protease inhibitors G. D. SEARLE & CO. (US) 1997-12-16 US disclosed
US-5510349-A HUMAN IMMUNODEFICIENCY VIRUS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510487-A TREATING HUMAN IMMUNODEFICIENCY VIRUS INFECTIONS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5510378-A Retroviral protease inhibitors G.D. SEARLE & CO. (US) 1996-04-23 US disclosed