SCHEMBL8734794

SCHEMBL8734794

O=C(Nc1cc(Cl)cc([N+](=O)[O-])c1NC(=O)C(F)(F)F)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 3/20 0.40
PDK2 Q15119 3/20 0.40
PDK3 Q15120 3/20 0.40
PDK4 Q16654 3/20 0.40
APP P05067 1/20 0.39
KCNMA1 Q12791 2/20 0.38
AR P10275 2/20 0.38
CYP3A4 P08684 2/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
HIF1A Q16665 1/20 0.37
TXNRD1 Q16881 1/20 0.37
TXNRD3 Q86VQ6 1/20 0.37
TXNRD2 Q9NNW7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
EPAS1 Q99814 1/20 0.36
PHGDH O43175 1/20 0.36
PGR P06401 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8734657 0.87 PDK1 (0.38) PDK1PDK2PDK3PDK4APP
SCHEMBL8736796 0.84 ALDH1A1 (0.40) PDK1PDK2PDK3PDK4APP
SCHEMBL16198090 0.83 KCNMA1 (0.38) APPKCNMA1CYP3A4ALDH1A1HPGD
SCHEMBL8734159 0.83 MAPK1 (0.48) KCNMA1ARCYP3A4ALDH1A1HPGD
SCHEMBL8936699 0.81 MAPT (0.51) PDK1PDK2PDK3PDK4APP
SCHEMBL8736871 0.80 ALDH1A1 (0.46) KCNMA1CYP3A4ALDH1A1HPGDALOX15
SCHEMBL8733248 0.78 MAPK1 (0.44) PDK1PDK2PDK3PDK4KCNMA1
SCHEMBL7784821 0.77 HRAS (0.41) PDK1PDK2PDK3PDK4KCNMA1
SCHEMBL7786526 0.76 CYP3A4 (0.40) PDK1PDK2PDK3PDK4AR
SCHEMBL11849607 0.76 ALDH1A1 (0.53) KCNMA1CYP3A4ALDH1A1HPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821953-A2 Anticoccidial methods and feedstuffs ELI LILLY AND COMPANY (US) 1998-02-04 EP disclosed