SCHEMBL8736796

SCHEMBL8736796

Nc1c(NC(=O)C(F)(F)F)cc(Cl)cc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
PDK1 Q15118 3/20 0.40
PDK2 Q15119 3/20 0.40
PDK3 Q15120 3/20 0.40
PDK4 Q16654 3/20 0.40
APP P05067 1/20 0.39
KCNMA1 Q12791 2/20 0.38
AR P10275 2/20 0.37
CYP3A4 P08684 2/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
HIF1A Q16665 1/20 0.36
TXNRD1 Q16881 1/20 0.36
TXNRD3 Q86VQ6 1/20 0.36
TXNRD2 Q9NNW7 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8736070 0.87 PDK1 (0.37) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL8734794 0.84 PDK1 (0.40) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL8736207 0.83 ALDH1A1 (0.57) ALDH1A1KCNMA1ARCYP3A4HPGD
SCHEMBL11404398 0.81 APP (0.41) ALDH1A1APPKCNMA1CYP3A4LMNA
SCHEMBL8936699 0.80 MAPT (0.51) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL1800375 0.75 PDK1 (0.42) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL16198090 0.74 KCNMA1 (0.38) ALDH1A1APPKCNMA1CYP3A4HPGD
SCHEMBL11850749 0.74 ALDH1A1 (0.37) ALDH1A1CYP3A4TSHREPAS1
SCHEMBL13592935 0.73 CXCR2 (0.46) ALDH1A1PDK1PDK2PDK3PDK4
SCHEMBL8736181 0.73 ALDH1A1 (0.55) ALDH1A1PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821953-A2 Anticoccidial methods and feedstuffs ELI LILLY AND COMPANY (US) 1998-02-04 EP disclosed