SCHEMBL873871

SCHEMBL873871

CC(C)CCNC(=O)c1ccc(-c2ccc(NC(=O)c3cc4cccnc4s3)cc2)o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
KDM4E B2RXH2 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
ALDH1A1 P00352 3/20 0.42
HSD17B10 Q99714 3/20 0.42
GAA P10253 3/20 0.42
HPGD P15428 2/20 0.42
NAMPT P43490 2/20 0.39
MAPK1 P28482 3/20 0.38
POLB P06746 2/20 0.38
MGAM O43451 2/20 0.38
SI P14410 2/20 0.38
MGAM2 Q2M2H8 2/20 0.38
PTPN1 P18031 1/20 0.38
PTPN11 Q06124 1/20 0.38
MAPT P10636 6/20 0.38
LMNA P02545 2/20 0.38
TP53 P04637 2/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874184 0.89 NPC1 (0.41) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL874680 0.87 NPC1 (0.46) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL873865 0.83 NAMPT (0.42) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL874535 0.83 NAMPT (0.48) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL874187 0.82 NPC1 (0.46) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL873905 0.81 DRD2 (0.48) ALDH1A1NAMPTCHRNA7
SCHEMBL874022 0.81 CHRNA7 (0.41) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL873709 0.81 CHRNA7 (0.41) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL874185 0.81 NPC1 (0.39) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL874135 0.81 NAMPT (0.41) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed