SCHEMBL873709

SCHEMBL873709

COC1CCN(CCNC(=O)c2ccc(-c3ccc(NC(=O)c4cc5cccnc5s4)cc3)o2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.41
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
NAMPT P43490 2/20 0.40
RXFP1 Q9HBX9 1/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPKAPK2 P49137 1/20 0.38
MEN1 O00255 1/20 0.38
APAF1 O14727 1/20 0.38
MAPK1 P28482 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874022 0.92 CHRNA7 (0.41) CHRNA7DRD2DRD3NAMPTRXFP1
SCHEMBL874535 0.89 NAMPT (0.48) CHRNA7DRD2DRD3NAMPTALDH1A1
SCHEMBL874135 0.86 NAMPT (0.41) CHRNA7DRD2DRD3NAMPTALDH1A1
SCHEMBL873905 0.84 DRD2 (0.48) CHRNA7DRD2DRD3NAMPTALDH1A1
SCHEMBL873710 0.83 CHRNA7 (0.41) CHRNA7NAMPTALDH1A1SMN1; SMN2MAPKAPK2
SCHEMBL873865 0.82 NAMPT (0.42) CHRNA7NAMPTALDH1A1SMN1; SMN2BCHE
SCHEMBL873871 0.81 NPC1 (0.42) CHRNA7NAMPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL874187 0.81 NPC1 (0.46) CHRNA7ALDH1A1SMN1; SMN2MEN1MAPK1
SCHEMBL874184 0.79 NPC1 (0.41) CHRNA7NAMPTRXFP1ALDH1A1SMN1; SMN2
SCHEMBL874680 0.78 NPC1 (0.46) ALDH1A1SMN1; SMN2MEN1MAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038905-A1 THIENOPYRIDINE NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed