SCHEMBL8742259

SCHEMBL8742259

COc1cc2ccc(CC(=S)N3CCOCC3)cc2cc1OC

nearest known ligand 0.79

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.79
MEN1 O00255 1/20 0.79
CYP2C19 P33261 1/20 0.79
ALDH1A1 P00352 11/20 0.67
HPGD P15428 5/20 0.67
MAPT P10636 4/20 0.67
GAA P10253 1/20 0.67
APOBEC3G Q9HC16 1/20 0.67
FAAH O00519 3/20 0.57
MGLL Q99685 3/20 0.57
HTT P42858 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.52
KDM4E B2RXH2 1/20 0.50
NQO1 P15559 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11277440 0.85 HTT (0.79) KMT2AMEN1CYP2C19ALDH1A1HPGD
SCHEMBL11274517 0.83 KMT2A (0.64) KMT2AMEN1CYP2C19ALDH1A1HPGD
SCHEMBL23048477 0.82 MGLL (0.65) KMT2AMEN1CYP2C19ALDH1A1HPGD
SCHEMBL4394405 0.81 ALDH1A1 (1.00) KMT2AMEN1CYP2C19ALDH1A1HPGD
SCHEMBL21455291 0.79 ALDH1A1 (0.71) KMT2AMEN1CYP2C19ALDH1A1HPGD
SCHEMBL11156037 0.74 MEN1 (0.67) KMT2AMEN1CYP2C19ALDH1A1HPGD
SCHEMBL9729243 0.74 MEN1 (0.63) KMT2AMEN1CYP2C19ALDH1A1HPGD
Hydrochloric Acid SCHEMBL11276469 0.74 SIGMAR1 (0.54) ALDH1A1HTTSMN1; SMN2
SCHEMBL4397261 0.73 ALDH1A1 (1.00) KMT2AMEN1CYP2C19ALDH1A1HPGD
SCHEMBL11277514 0.72 HTT (0.60) KMT2AMEN1ALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618822-A N-substituted trifluoromethylphenyltetrahydropyridines, process for the preparation thereof, intermediates in said process and pharmaceutical compositions containing them SANOFI (FR) 1997-04-08 US disclosed
US-5599941-A N-substituted trifluoromethylphenyltetrahydropyridines process for the preparation thereof intermediates in said process and pharmaceutical compositions containing them SANOFI (FR) 1997-02-04 US disclosed
US-5596101-A N-substituted trifluoromethylphenyltetrahydropyridines, process for the preparation thereof, intermediates in said process and pharmaceutical compositions containing them SANOFI (FR) 1997-01-21 US disclosed
US-5559238-A N-substituted trifluoromethylphenyltetrahydropyridenes process for the preparation thereof, intermediates in said process and pharmaceutical compositions containing them SANOFI (FR) 1996-09-24 US disclosed
US-5462945-A N-substituted trifluoromethylphenyltetrahydropyridines, process for the preparation thereof, intermediates in said process and pharmaceutical compositions containing them SANOFI (FR) 1995-10-31 US disclosed
EP-0458697-B1 N-substituted trifluoromethylphenyl tetrahydropyridines, process for their preparation, intermediates and pharmaceutical preparations containing them SANOFI ELF (FR) 1994-07-27 EP disclosed
US-5281606-A N-substituted trifluoromethylphenyltetrahydropyridines, process for the preparation thereof, intermediates in said process and pharmaceutical compositions containing them SANOFI (FR) 1994-01-25 US disclosed
EP-0458697-A1 N-substituted trifluoromethylphenyl tetrahydropyridines, process for their preparation, intermediates and pharmaceutical preparations containing them ELF SANOFI (FR) 1991-11-27 EP disclosed
US-4327022-A Heterocyclic alkyl naphthols STERLING DRUG INC. (US) 1982-04-27 US disclosed
US-4169108-A 5(OR 6)-[(Substituted-amino)alkyl]-2,3-naphthalenediols STERLING DRUG INC. (US) 1979-09-25 US disclosed