SCHEMBL8743012

SCHEMBL8743012

[CH2]OC(=O)N1CCNCC1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA9 Q16790 1/20 0.48
CHKA P35790 1/20 0.46
CHRNB2 P17787 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
CHRNB3 Q05901 1/20 0.45
CHRNA6 Q15825 1/20 0.45
TPSAB1 Q15661 1/20 0.40
TPSD1 Q9BZJ3 1/20 0.40
TPSG1 Q9NRR2 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
HSD11B1 P28845 1/20 0.38
POLB P06746 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
EPHX2 P34913 1/20 0.35
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4341361 0.80 CA2 (0.43) CA2CA12CA1CA9CHKA
SCHEMBL8103057 0.80 CHRNB2 (0.54) CA2CA12CA1CA9CHKA
SCHEMBL3635077 0.77
SCHEMBL316937 0.76 CHRNB2 (0.50) CA2CA12CA1CA9CHKA
SCHEMBL20369074 0.76 CA2 (0.48) CA2CA12CA1CA9CHKA
SCHEMBL6721 0.76 CHRNB2 (0.50) CA2CA12CA1CA9CHKA
SCHEMBL1780077 0.76 LMNA (0.43) CA2CA12CA1CA9CHKA
SCHEMBL304390 0.75 ALDH1A1 (0.50) CA2CHKAHSD11B1POLBHPGD
Ethane SCHEMBL27604108 0.74 CHRNB2 (0.48) CA2CA12CA1CA9CHKA
SCHEMBL28744445 0.74 CHRNB2 (0.48) CA2CA12CA1CA9CHKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354913-A Chemical intermediates for drugs or drugs as thromboxane, prostaglandin antagonist, lipoxygenase enzyme inhibitor, antioxidants TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US claimed
EP-0751113-A1 Optically active phenol derivatives and preparation thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-02 EP disclosed
EP-0537954-B1 Process of preparing diphenylmethane derivatives TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-07-24 EP disclosed
US-5420363-A Catalytic reaction of phenol with secondary carbinol for enantiomorphs TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-05-30 US disclosed
US-5354913-A Chemical intermediates for drugs or drugs as thromboxane, prostaglandin antagonist, lipoxygenase enzyme inhibitor, antioxidants TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed
EP-0582382-A2 Optically active phenol derivatives and preparation thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-02-09 EP disclosed
EP-0295037-B1 PHENOL DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-08-18 EP disclosed
US-5235091-A Reacting a phenol compound with a stilbene compound in presence of methanesulfonic acid TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-08-10 US disclosed
EP-0537954-A1 Process of preparing diphenylmethane derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-04-21 EP disclosed
US-5162571-A Phenol derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-11-10 US disclosed
EP-0295037-A2 Phenol derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-12-14 EP disclosed