SCHEMBL874741

SCHEMBL874741

O=C(NC1CC1)c1sc(-c2ccc([N+](=O)[O-])cc2)nc1-c1ccsc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 2/20 0.47
HPGD P15428 1/20 0.47
RAB9A P51151 1/20 0.46
PPARA Q07869 2/20 0.45
POLB P06746 1/20 0.41
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
CSNK2A1 P68400 1/20 0.38
IDH2 P48735 1/20 0.38
APP P05067 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
CDC7 O00311 2/20 0.38
DBF4 Q9UBU7 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL874429 0.85 CDC7 (0.42) ALDH1A1MAPTRAB9ACDC7DBF4
SCHEMBL874800 0.83 RAB9A (0.62) KMT2ASMN1; SMN2MEN1ALDH1A1MAPT
SCHEMBL874757 0.71 HDAC1 (0.44)
SCHEMBL30583813 0.67 NPC1 (0.57) KMT2ASMN1; SMN2MEN1ALDH1A1MAPT
SCHEMBL28975685 0.67 NPC1 (0.57) KMT2ASMN1; SMN2MEN1ALDH1A1MAPT
SCHEMBL30583812 0.67 NPC1 (0.57) KMT2ASMN1; SMN2MEN1ALDH1A1MAPT
SCHEMBL24726553 0.66 APP (0.52) ALDH1A1MAPTRAB9APOLBAPP
SCHEMBL18458068 0.66 POLB (0.56) KMT2ASMN1; SMN2MEN1ALDH1A1MAPT
SCHEMBL10909889 0.66 MAPT (0.62) KMT2ASMN1; SMN2MEN1ALDH1A1MAPT
SCHEMBL874528 0.64 RAB9A (0.72) KMT2ASMN1; SMN2MEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038904-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-03-29 WO disclosed