SCHEMBL8744771

SCHEMBL8744771

CCOC(=O)[C@H](C)N(C)C(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.46
AKR1B1 P15121 1/20 0.45
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 4/20 0.43
MEN1 O00255 2/20 0.43
NPC1 O15118 1/20 0.43
HTT P42858 2/20 0.42
CASP1 P29466 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
KDM4E B2RXH2 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
ALOX15 P16050 1/20 0.40
NLRP3 Q96P20 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9368074 0.87 RORC (0.46) RORCAKR1B1ALDH1A1KMT2AMEN1
SCHEMBL9319221 0.86 CASP1 (0.47) RORCAKR1B1ALDH1A1KMT2AMEN1
SCHEMBL9319501 0.83 AKR1B1 (0.44) AKR1B1ALDH1A1KMT2AMEN1NPC1
SCHEMBL9321052 0.83 UTS2R (0.42) AKR1B1ALDH1A1KMT2AMEN1NPC1
SCHEMBL9482977 0.82 RORC (0.42) RORCAKR1B1ALDH1A1KMT2AMEN1
SCHEMBL9319787 0.82 AKR1B1 (0.40) RORCAKR1B1ALDH1A1KMT2AMEN1
SCHEMBL9318635 0.81 ALDH1A1 (0.39) AKR1B1ALDH1A1KMT2AMEN1NPC1
SCHEMBL9319168 0.80 EPHX2 (0.41) RORCAKR1B1ALDH1A1KMT2AMEN1
SCHEMBL9321062 0.80 C5AR1 (0.42) RORCAKR1B1ALDH1A1KMT2AMEN1
SCHEMBL9373305 0.80 RORC (0.41) RORCAKR1B1ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
EP-0377893-B1 3-Aryl-pyrrolidine-2,4-dione derivatives BAYER AG (DE) 1994-04-06 EP disclosed
US-5186737-A Herbicides BAYER AKTIENGESELLSCHAFT (DE) 1993-02-16 US disclosed
US-5045560-A Insecticides, nematocides, fungicides, herbicides, human and veterinary medicine BAYER AKTIENGESELLSCHAFT (DE) 1991-09-03 US disclosed
EP-0377893-A2 3-Aryl-pyrrolidine-2,4-dione derivatives BAYER AG (DE) 1990-07-18 EP disclosed