SCHEMBL874517

SCHEMBL874517

CCCOc1ccccc1C(=O)N1C[C@@H](N(C)C)C[C@H]1C(=O)Nc1ccc(CCc2ccc(NC(=O)[C@@H]3C[C@H](N(C)C)CN3)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.36
TP53 P04637 1/20 0.36
CFTR P13569 14/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845092 0.92 TP53 (0.41) THRBTP53CFTR
SCHEMBL13272447 0.84 BCHE (0.31) CFTR
SCHEMBL873764 0.84 TP53 (0.35) THRBTP53CFTR
SCHEMBL845096 0.83 TP53 (0.40) THRBTP53
SCHEMBL873619 0.76 TP53 (0.34) THRBTP53
SCHEMBL845370 0.69 PIK3CA (0.37) THRB
SCHEMBL845518 0.66 GAA (0.52) TP53
SCHEMBL845354 0.61 POLB (0.57) TP53
SCHEMBL872930 0.60 GAA (0.52)
SCHEMBL17502615 0.59 NPSR1 (0.60) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed