SCHEMBL845096

SCHEMBL845096

CCCOc1ccccc1C(=O)N1C[C@@H](N(C)C)C[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C[C@H](N(C)C)CN3C(=O)c3ccccc3OCCC)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.40
GAA P10253 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
TSHR P16473 1/20 0.35
THRB P10828 1/20 0.35
PNLIP P16233 1/20 0.35
PIK3CA P42336 2/20 0.34
MTOR P42345 2/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MCL1 Q07820 1/20 0.34
MRGPRX1 Q96LB2 1/20 0.34
AGTR2 P50052 1/20 0.34
HIF1A Q16665 1/20 0.34
FAAH O00519 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873619 0.91 TP53 (0.34) TP53GAAMEN1KMT2ATSHR
SCHEMBL845092 0.90 TP53 (0.41) TP53THRB
SCHEMBL845370 0.85 PIK3CA (0.37) MEN1KMT2ATHRBPIK3CAMTOR
SCHEMBL874517 0.83 THRB (0.36) TP53THRB
SCHEMBL873764 0.82 TP53 (0.35) TP53THRB
SCHEMBL845518 0.82 GAA (0.52) TP53GAAMEN1KMT2ATSHR
SCHEMBL872515 0.79 PIK3CA (0.33) MEN1KMT2ATHRBPIK3CAMTOR
SCHEMBL845439 0.79 ALDH1A1 (0.38) MEN1KMT2APIK3CAMTORPIK3CD
SCHEMBL845429 0.76 CTSS (0.44) MEN1KMT2AALDH1A1
SCHEMBL845354 0.75 POLB (0.57) TP53MEN1KMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed