SCHEMBL873619

SCHEMBL873619

CCCOc1ccccc1CON1C[C@@H](N(C)C)C[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C[C@H](N(C)C)CN3C(=O)c3ccccc3OCCC)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.34
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
ALDH1A1 P00352 1/20 0.31
MCL1 Q07820 1/20 0.31
GAA P10253 1/20 0.31
HCRTR1 O43613 1/20 0.30
HCRTR2 O43614 1/20 0.30
THRB P10828 1/20 0.30
PIK3CA P42336 2/20 0.30
MTOR P42345 2/20 0.30
PIK3CD O00329 1/20 0.30
PIK3CB P42338 1/20 0.30
PIK3CG P48736 1/20 0.30
MEN1 O00255 1/20 0.30
TSHR P16473 1/20 0.30
KMT2A Q03164 1/20 0.30
PNLIP P16233 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873764 0.92 TP53 (0.35) TP53HCRTR1HCRTR2THRB
SCHEMBL845096 0.91 TP53 (0.40) TP53ALDH1A1MCL1GAATHRB
SCHEMBL872515 0.87 PIK3CA (0.33) THRBPIK3CAMTORPIK3CDPIK3CB
SCHEMBL845092 0.82 TP53 (0.41) TP53THRB
SCHEMBL845370 0.81 PIK3CA (0.37) HCRTR1HCRTR2THRBPIK3CAMTOR
SCHEMBL10119511 0.81 GAA (0.44) TP53ALDH1A1GAAMEN1TSHR
SCHEMBL872636 0.81 POLB (0.33) BCHEACHEALDH1A1PIK3CAMTOR
SCHEMBL874517 0.76 THRB (0.36) TP53THRB
SCHEMBL845518 0.74 GAA (0.52) TP53ALDH1A1GAAMEN1TSHR
SCHEMBL873095 0.72 HDAC8 (0.38) BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed