SCHEMBL8745816

SCHEMBL8745816

CCOc1cc2c(C)c(CCN3CCN(c4ccccc4OC)CC3)c(=O)oc2cc1OC

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.55
ADRA1D P25100 3/20 0.55
ADRA1B P35368 3/20 0.55
DRD2 P14416 2/20 0.51
BRAF P15056 1/20 0.51
HTR2A P28223 1/20 0.51
KCNH2 Q12809 1/20 0.50
GAA P10253 1/20 0.49
DRD3 P35462 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745798 0.94 BRAF (0.56) ADRA1AADRA1DADRA1BDRD2BRAF
SCHEMBL9144743 0.93 DRD2 (0.51) ADRA1ADRD2BRAFHTR2AKCNH2
SCHEMBL8745782 0.90 DRD2 (0.54) ADRA1AADRA1DADRA1BDRD2BRAF
SCHEMBL8745813 0.89 BRAF (0.49) ADRA1AADRA1DADRA1BDRD2BRAF
SCHEMBL8745760 0.89 ADRA1A (0.55) ADRA1AADRA1DADRA1BDRD2BRAF
SCHEMBL8745769 0.87 BRAF (0.55) ADRA1AADRA1DADRA1BDRD2BRAF
SCHEMBL8745809 0.84 HTR2A (0.60) ADRA1ADRD2BRAFHTR2AKCNH2
SCHEMBL8745781 0.84 ADRA1A (0.51) ADRA1AADRA1DADRA1BDRD2HTR2A
SCHEMBL8745759 0.84 DRD2 (0.59) DRD2BRAFHTR2AKCNH2DRD3
Ensaculin SCHEMBL29722503 0.83 HTR2A (0.63) ADRA1ADRD2HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed