SCHEMBL8745813

SCHEMBL8745813

CCS(=O)(=O)Oc1cc2c(C)c(CCN3CCN(c4ccccc4OC)CC3)c(=O)oc2cc1OC

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.49
DRD2 P14416 4/20 0.47
ADRA1A P35348 2/20 0.47
HTR2A P28223 1/20 0.47
GAA P10253 1/20 0.47
KCNH2 Q12809 1/20 0.46
DRD3 P35462 2/20 0.46
ADRA1D P25100 1/20 0.45
ADRA1B P35368 1/20 0.45
HTR1A P08908 1/20 0.45
NTSR1 P30989 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745798 0.92 BRAF (0.56) BRAFDRD2ADRA1AHTR2AGAA
SCHEMBL8745816 0.89 ADRA1A (0.55) BRAFDRD2ADRA1AHTR2AGAA
SCHEMBL9144743 0.87 DRD2 (0.51) BRAFDRD2ADRA1AHTR2AKCNH2
SCHEMBL8745760 0.86 ADRA1A (0.55) BRAFDRD2ADRA1AHTR2AGAA
SCHEMBL8745769 0.85 BRAF (0.55) BRAFDRD2ADRA1AHTR2AGAA
SCHEMBL8745809 0.82 HTR2A (0.60) BRAFDRD2ADRA1AHTR2AKCNH2
SCHEMBL8745759 0.82 DRD2 (0.59) BRAFDRD2HTR2AKCNH2DRD3
SCHEMBL8745782 0.79 DRD2 (0.54) BRAFDRD2ADRA1AHTR2AKCNH2
Ensaculin SCHEMBL29722503 0.78 HTR2A (0.63) DRD2ADRA1AHTR2AKCNH2HTR1A
Ensaculin SCHEMBL677971 0.78 HTR2A (0.63) DRD2ADRA1AHTR2AKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0663911-B1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE SCHWABE WILLMAR GMBH & CO (DE) 1997-02-05 EP disclosed
US-5550129-A THERAPY FOR NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS WILLMAR SCHWABE GMBH & CO. (DE) 1996-08-27 US disclosed
EP-0663911-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE. SCHWABE WILLMAR GMBH & CO (DE) 1995-07-26 EP disclosed
WO-1994008985-A1 BENZOPYRANONES, METHOD OF PREPARING THEM AND THEIR USE DR. WILLMAR SCHWABE GMBH & CO. (DE) 1994-04-28 WO disclosed