SCHEMBL8747860

SCHEMBL8747860

OC12CCC(c3ccc(CBr)cc3)(CC1)CC2

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
PNMT P11086 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9250332 0.76 CA2 (0.47) ALDH1A1TSHR
SCHEMBL15524912 0.73 HRH3 (0.41) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL29268172 0.70 TRPA1 (0.40) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL5280539 0.68 LMNA (0.57) ALDH1A1
SCHEMBL22027005 0.67 LMNA (0.54)
SCHEMBL14166006 0.67 AKR1C1 (0.50) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL131361 0.66 ALDH1A1 (0.67) TRPA1ALDH1A1TSHRCES2CES1
SCHEMBL4680071 0.64 AKR1C1 (0.61) TSHRCES2CES1
SCHEMBL12982189 0.64 TSHR (0.34) TRPA1ALDH1A1TSHR
SCHEMBL118612 0.64 OPRM1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0599732-B1 Derivatives of 1-phenylbicyclo-2,2,2-octane, their preparation process and pharmaceutical compositions containing them ADIR (FR) 1997-03-12 EP disclosed
US-5403953-A Antiarthritic and -inflammatory agents ADIR ET COMPAGNIE (FR) 1995-04-04 US disclosed
EP-0599732-A1 Derivatives of 1-phenylbicyclo-2,2,2-octane, their preparation process and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-06-01 EP disclosed