SCHEMBL8750890

SCHEMBL8750890

CC(=O)OC(NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSL P07711 9/20 0.62
CTSB P07858 4/20 0.62
CTSS P25774 2/20 0.62
CTSK P43235 2/20 0.62
TACR1 P25103 2/20 0.60
ALDH1A1 P00352 1/20 0.58
ALOX15 P16050 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8750936 0.94 CTSL (0.61) CTSLCTSBCTSSCTSKTACR1
SCHEMBL10861784 0.87 ALDH1A1 (0.56) CTSLCTSBCTSSCTSKALDH1A1
SCHEMBL10607439 0.85 CTSK (0.55) CTSLCTSBCTSSCTSKALDH1A1
SCHEMBL12952246 0.84 CTSL (0.69) CTSLCTSBCTSSCTSKTACR1
SCHEMBL8668091 0.83 TACR1 (0.70) CTSLCTSBCTSSCTSKTACR1
SCHEMBL7268361 0.83 CTSL (0.65) CTSLCTSBCTSSCTSKTACR1
SCHEMBL19807564 0.82 TACR1 (0.72) CTSLCTSBCTSSCTSKTACR1
SCHEMBL10802556 0.82 CTSL (0.70) CTSLCTSBCTSSCTSKTACR1
SCHEMBL7268180 0.81 TACR1 (0.64) CTSLCTSBCTSSCTSKTACR1
SCHEMBL9725868 0.81 CTSL (0.60) CTSLCTSBCTSSCTSKTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0561303-B1 Conjugates of phenylalanine-glycine with antitumor substances KUREHA CHEMICAL IND CO LTD (JP) 1997-02-26 EP disclosed
US-5470960-A Antitumor agents KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-11-28 US disclosed
US-5411964-A Phenylalanine-glycine compounds having anti-tumor activity, process for preparation thereof, and pharmaceutical composition containing said compounds KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1995-05-02 US disclosed
EP-0561303-A2 Conjugates of phenylalanine-glycine with antitumor substances KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 1993-09-22 EP disclosed