SCHEMBL875341

SCHEMBL875341

N[C@@H]1COc2cccc(O)c2C1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.45
DRD3 P35462 1/20 0.45
DPP4 P27487 1/20 0.44
DYRK1A Q13627 1/20 0.35
NISCH Q9Y2I1 1/20 0.34
ALOX15B O15296 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
MAOA P21397 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30601522 1.00 DRD2 (0.45) DRD2DRD3DPP4DYRK1ANISCH
SCHEMBL9392163 1.00 DRD2 (0.45) DRD2DRD3DPP4DYRK1ANISCH
SCHEMBL21585684 0.80 DPP4 (0.39) DRD2DRD3DPP4DYRK1AALOX15B
SCHEMBL9900909 0.79 MAOA (0.40) DRD2DRD3DPP4MAOA
SCHEMBL23652957 0.79 AADAT (0.37) DPP4
SCHEMBL19054489 0.79 HTR7 (0.38) DRD2
SCHEMBL10699275 0.79 DRD2 (0.33) DRD2
Hydrochloric Acid SCHEMBL21810859 0.77 HTR2A (0.34) DRD2
SCHEMBL5761600 0.77 PARP1 (0.43) DRD2
SCHEMBL8854697 0.76 MEN1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012039657-A1 NOVEL CHROMANE COMPOUND FOR THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2012-03-29 WO disclosed
WO-2012039657-A1 NOVEL CHROMANE COMPOUND FOR THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2012-03-29 WO disclosed