SCHEMBL876160

SCHEMBL876160

CN(C(=O)c1ccc2c(c1)C(N1C=C(OC(=O)O)C(C(F)(F)F)=CC1)CCO2)C1CCN(c2ccncc2)CC1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
F10 P00742 4/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CCR5 P51681 1/20 0.32
MCHR1 Q99705 2/20 0.31
SMO Q99835 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL876437 0.88 F10 (0.33) F10CCR5MCHR1
SCHEMBL876499 0.87 SLC2A1 (0.35) F10CCR5MCHR1
SCHEMBL875680 0.86 F10 (0.33) F10CCR5MCHR1
SCHEMBL876268 0.80 F10 (0.34) F10NPC1RAB9ACCR5MCHR1
SCHEMBL878327 0.79 TLR9 (0.36) F10
SCHEMBL876159 0.78 NPC1 (0.35) F10NPC1RAB9ACCR5MCHR1
SCHEMBL876267 0.78 F10 (0.36) F10NPC1RAB9ACCR5
SCHEMBL784870 0.75 F10 (0.42) F10NPC1RAB9ACCR5
SCHEMBL784756 0.72 F10 (0.40) F10NPC1RAB9ACCR5
SCHEMBL876778 0.72 BDKRB1 (0.39) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed