SCHEMBL8764359

SCHEMBL8764359

N#Cc1ccc(S(=O)(=O)CS(=O)(=O)C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
CYP19A1 P11511 2/20 0.42
NR1I2 O75469 1/20 0.39
RORA P35398 1/20 0.39
RORC P51449 1/20 0.39
NR1H2 P55055 1/20 0.39
RORB Q92753 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
ALDH1A1 P00352 1/20 0.39
NR1H3 Q13133 1/20 0.39
KIF11 P52732 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
TRPV4 Q9HBA0 1/20 0.37
PLCG1 P19174 1/20 0.37
KDM1A O60341 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8763331 0.78 ALDH1A1 (0.43) CA1CA2ALDH1A1PLCG1
SCHEMBL8764344 0.77 MMP1 (0.49) MAPTCA12CA1CA2CA9
SCHEMBL8764317 0.77 PLCG1 (0.67) MAPTCA12CA1CA2CA9
SCHEMBL6855152 0.77 ALDH1A1 (0.52) MAPTCA12CA1CA2CA9
SCHEMBL8764352 0.77 NPC1 (0.46) CA12CA1CA2CA9ALDH1A1
SCHEMBL2325842 0.76 CA1 (0.50) CA12CA1CA2CA9CYP19A1
SCHEMBL8764400 0.76 PSIP1 (0.50) CA12CA1CA2CA9ALDH1A1
SCHEMBL506270 0.74 MAPT (0.55) MAPTCA12CA1CA2CA9
SCHEMBL13363525 0.73 EPAS1 (0.49) CA12CA1CA2CA9CYP19A1
SCHEMBL8763322 0.72 CA1 (0.47) CA12CA1CA2CA9RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0606756-B1 Use of disulfonyl methanes for the control of parasites LILLY CO ELI (US) 1997-07-23 EP disclosed
US-5614525-A ANTHELMINTICS ELI LILLY AND COMPANY (US) 1997-03-25 US disclosed
US-5596122-A INSECTICIDES AND LARVICIDES ELI LILLY AND COMPANY (US) 1997-01-21 US disclosed
US-5449681-A Administering by mouth or injection; anthelmintics, insecticides ELI LILLY AND COMPANY (US) 1995-09-12 US disclosed
EP-0606756-A1 Use of disulfonyl methanes for the control of parasites ELI LILLY AND COMPANY (US) 1994-07-20 EP disclosed