SCHEMBL876499

SCHEMBL876499

CN(C(=O)c1ccc2c(c1)C(N1C=C(OC(=O)O)C(C(F)(F)F)=CC1)CCC2)C1CCN(c2ccncc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 2/20 0.35
PDK2 Q15119 1/20 0.33
POLB P06746 1/20 0.32
F10 P00742 4/20 0.32
MCHR1 Q99705 1/20 0.32
CCR5 P51681 1/20 0.32
JAK2 O60674 3/20 0.31
JAK1 P23458 3/20 0.31
GPR55 Q9Y2T6 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL876437 0.96 F10 (0.33) SLC2A1PDK2POLBF10MCHR1
SCHEMBL875680 0.90 F10 (0.33) SLC2A1PDK2F10MCHR1CCR5
SCHEMBL876160 0.87 F10 (0.33) F10MCHR1CCR5
SCHEMBL878327 0.86 TLR9 (0.36) PDK2F10JAK2JAK1
SCHEMBL876131 0.80 POLB (0.34) SLC2A1POLBF10MCHR1CCR5
SCHEMBL876715 0.80 CCR5 (0.37) PDK2POLBF10MCHR1CCR5
SCHEMBL876778 0.80 BDKRB1 (0.39) F10
SCHEMBL876498 0.78 SLC2A1 (0.38) SLC2A1PDK2POLBF10MCHR1
SCHEMBL876130 0.77 POLB (0.35) SLC2A1POLBF10MCHR1CCR5
SCHEMBL878508 0.75 F10 (0.34) POLBF10MCHR1CCR5JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed