SCHEMBL8766342

SCHEMBL8766342

CCCc1ccc(-c2cc(F)c(C#Cc3ccc(F)c(F)c3)c(F)c2)nc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.54
RAB9A P51151 7/20 0.54
NPC1 O15118 6/20 0.54
TP53 P04637 3/20 0.54
PKM P14618 1/20 0.54
HSD17B10 Q99714 1/20 0.54
NFKB1 P19838 3/20 0.40
NFKB2 Q00653 3/20 0.40
RELA Q04206 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAPK1 P28482 2/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
MAPT P10636 4/20 0.39
KDM4E B2RXH2 1/20 0.38
MITF O75030 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
KLF5 Q13887 1/20 0.38
THRB P10828 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766676 0.93 RAB9A (0.50) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL8766722 0.92 RAB9A (0.49) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL9434295 0.90 NPC1 (0.41) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL9433719 0.90 SMN1; SMN2 (0.48) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL8766807 0.85 RAB9A (0.39) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL8767583 0.85 NPC1 (0.39) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL9433261 0.83 RAB9A (0.47) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL9433608 0.82 RAB9A (0.46) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL8766245 0.82 ALDH1A1 (0.41) SMN1; SMN2RAB9ANPC1TP53PKM
SCHEMBL8766258 0.82 CYP17A1 (0.37) SMN1; SMN2RAB9ANPC1TP53PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543244-B1 Fluoro substituted tolans and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 1997-08-20 EP disclosed
US-5372746-A Fluoro-substituted tolane compounds and liquid crystalline mixtures containing same HOFFMANN-LA ROCHE INC. (US) 1994-12-13 US disclosed
EP-0543244-A1 Fluoro substituted tolans and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed