SCHEMBL8766708

SCHEMBL8766708

C#CC(CCCc1ccco1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP3A4 P08684 1/20 0.49
ALOX15 P16050 1/20 0.49
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40
SLC1A1 P43005 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
USP2 O75604 2/20 0.39
HPGD P15428 1/20 0.39
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
HSD17B10 Q99714 1/20 0.38
EPHX2 P34913 3/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPN7 P35236 1/20 0.37
BLM P54132 1/20 0.37
KMT2A Q03164 1/20 0.37
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8765582 0.73 CYP2C19 (0.49) ALDH1A1SLC1A3SLC1A2SLC1A1TDP1
SCHEMBL28367950 0.72 ALDH1A1 (0.49) ALDH1A1CYP3A4ALOX15TDP1USP2
SCHEMBL27584268 0.71 POLB (0.47) ALDH1A1SLC1A3SLC1A2SLC1A1TDP1
Bicarbonate SCHEMBL29658892 0.71 ALDH1A1 (0.52) ALDH1A1CYP3A4ALOX15SLC1A3SLC1A2
SCHEMBL8765876 0.71 NAAA (0.35)
SCHEMBL2199125 0.71 MAPK1 (0.52) ALDH1A1CYP3A4ALOX15TDP1USP2
SCHEMBL9705770 0.69 MAPT (0.52) ALDH1A1CYP3A4ALOX15TDP1USP2
Hydrochloric Acid SCHEMBL11635247 0.69 MAPK1 (0.50) ALDH1A1CYP3A4ALOX15TDP1USP2
SCHEMBL16672942 0.69 ERAP1 (0.46) HPGDKMT2ATSHR
SCHEMBL7094868 0.69 ALDH1A1 (0.67) ALDH1A1CYP3A4ALOX15TDP1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1997-07-30 EP disclosed
WO-1996011686-A1 DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-04-25 WO disclosed