SCHEMBL8767110

SCHEMBL8767110

CCOC(=O)CNC(=O)Oc1ncc(C(=O)NS(=O)(=O)c2ccc(C(=O)NC3CCCCC3)cc2)cc1OCC(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.40
TSHR P16473 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTT P42858 2/20 0.40
BLM P54132 2/20 0.39
CYP3A4 P08684 1/20 0.39
HTR1A P08908 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
NFKB1 P19838 1/20 0.39
CNR1 P21554 1/20 0.39
CYP2C19 P33261 1/20 0.39
ADRA1A P35348 1/20 0.39
KMT2A Q03164 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
NR3C1 P04150 1/20 0.38
AR P10275 1/20 0.38
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8768279 0.91 LMNA (0.42) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8767453 0.91 LMNA (0.42) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8875248 0.89 LMNA (0.41) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8768228 0.86 LMNA (0.45) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8103313 0.86 LMNA (0.45) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8099449 0.85 LMNA (0.37) LMNASMN1; SMN2HTT
SCHEMBL8104049 0.83 LMNA (0.39) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8103050 0.82 LMNA (0.44) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8768360 0.82 L3MBTL1 (0.50) LMNATSHRSMN1; SMN2HTTBLM
SCHEMBL8874675 0.81 L3MBTL1 (0.43) LMNATSHRSMN1; SMN2HTTBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673931-B1 Sulfonamidocarbonyl-pyridine-2-carboxamides and their pyridine-N-oxides, process for their preparation and their use as medicaments HOECHST AG (DE) 1997-08-13 EP disclosed
EP-0673931-A1 Sulfonamidocarbonyl-pyridine-2-carboxamides and their pyridine-N-oxides, process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-09-27 EP disclosed