SCHEMBL8767188

SCHEMBL8767188

CCCCOc1ccc(-c2cc(F)c(C#Cc3ccc(F)c(F)c3)c(F)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.45
RARA P10276 1/20 0.45
CYP2D6 P10635 5/20 0.43
CYP3A4 P08684 3/20 0.43
CYP19A1 P11511 5/20 0.40
CYP2C9 P11712 5/20 0.40
CYP2C19 P33261 5/20 0.40
CYP1A2 P05177 4/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MCHR1 Q99705 2/20 0.39
CHRM1 P11229 1/20 0.39
HTR2A P28223 1/20 0.39
MCL1 Q07820 1/20 0.39
ERN1 O75460 1/20 0.38
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766249 0.96 RARA (0.41) RARBRARACYP2D6CYP3A4MCHR1
SCHEMBL8767150 0.89 CHRNA7 (0.41) NPC1RAB9ASMN1; SMN2MCHR1CHRM1
SCHEMBL9470533 0.86 GRM5 (0.44) RARBRARACYP2D6CYP3A4NPC1
SCHEMBL9434250 0.85 MCHR1 (0.40) RARBRARACYP2D6CYP3A4NPC1
SCHEMBL8767540 0.84 TSHR (0.43) RARBRARAHSD17B10ALDH1A1
SCHEMBL9469637 0.83 NR5A1 (0.47) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL8766681 0.83 HSD17B10 (0.49) RARBRARACYP3A4HSD17B10CHRM1
SCHEMBL9469740 0.83 ACACB (0.46)
SCHEMBL8767207 0.82 HSD17B10 (0.51) RARBRARACYP3A4RAB9ASMN1; SMN2
SCHEMBL8766844 0.82 HSD17B10 (0.51) RARBRARACYP3A4RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543244-B1 Fluoro substituted tolans and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 1997-08-20 EP disclosed
US-5372746-A Fluoro-substituted tolane compounds and liquid crystalline mixtures containing same HOFFMANN-LA ROCHE INC. (US) 1994-12-13 US disclosed
EP-0543244-A1 Fluoro substituted tolans and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed