SCHEMBL8766249

SCHEMBL8766249

CCCOc1ccc(-c2cc(F)c(C#Cc3ccc(F)c(F)c3)c(F)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RARA P10276 1/20 0.41
RARB P10826 1/20 0.41
ERN1 O75460 1/20 0.41
MCHR1 Q99705 2/20 0.40
CHRM1 P11229 1/20 0.40
HTR2A P28223 1/20 0.40
MAOB P27338 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
GRM5 P41594 1/20 0.38
ACACB O00763 9/20 0.37
MAOA P21397 1/20 0.37
ACACA Q13085 1/20 0.36
APP P05067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8767188 0.96 RARB (0.45) RARARARBERN1MCHR1CHRM1
SCHEMBL8767150 0.90 CHRNA7 (0.41) ERN1MCHR1CHRM1HTR2AGRM5
SCHEMBL9434250 0.88 MCHR1 (0.40) RARARARBERN1MCHR1CHRM1
SCHEMBL9469740 0.87 ACACB (0.46) GRM5ACACBAPP
SCHEMBL8766245 0.85 ALDH1A1 (0.41) MCHR1CHRM1HTR2ACYP2D6GRM5
SCHEMBL8766829 0.85 NPC1 (0.40) MCHR1CHRM1HTR2AGRM5ACACB
SCHEMBL9433854 0.83 MAOB (0.38) MCHR1CHRM1HTR2AMAOBCYP2D6
SCHEMBL8766258 0.82 CYP17A1 (0.37) RARARARBMAOBGRM5ACACB
SCHEMBL8766246 0.82 CYP17A1 (0.39) RARARARBGRM5ACACB
SCHEMBL9470533 0.81 GRM5 (0.44) RARARARBMCHR1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543244-B1 Fluoro substituted tolans and liquid crystal mixtures containing them MERCK PATENT GMBH (DE) 1997-08-20 EP disclosed
US-5372746-A Fluoro-substituted tolane compounds and liquid crystalline mixtures containing same HOFFMANN-LA ROCHE INC. (US) 1994-12-13 US disclosed
EP-0543244-A1 Fluoro substituted tolans and liquid crystal mixtures containing them F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed