SCHEMBL8768626

SCHEMBL8768626

C=CCc1ccc(-c2ccccc2)c(-c2ccc(C#N)c(F)c2F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.39
KDM4E B2RXH2 3/20 0.37
GAA P10253 3/20 0.37
ALDH1A1 P00352 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HPGD P15428 2/20 0.37
MEN1 O00255 2/20 0.37
MAPT P10636 2/20 0.37
GABRA1 P14867 2/20 0.37
CNR1 P21554 2/20 0.37
CNR2 P34972 2/20 0.37
GABRB2 P47870 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH2 P05091 1/20 0.37
AKR1B1 P15121 1/20 0.37
PPARG P37231 1/20 0.37
PPARD Q03181 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5573395 0.81 CYP19A1 (0.51) CYP19A1KDM4EGAAALDH1A1NPSR1
SCHEMBL7198375 0.78 GABRA1 (0.41) CYP19A1KDM4EGAAALDH1A1NPSR1
SCHEMBL4620939 0.78 GABRA1 (0.41) CYP19A1KDM4EGAAALDH1A1NPSR1
SCHEMBL27416538 0.76 EGLN2 (0.44) KDM4EGAAALDH1A1NPSR1HPGD
SCHEMBL9274282 0.75 GABRA1 (0.50) KDM4EGAAALDH1A1NPSR1HPGD
SCHEMBL29027369 0.74 GABRA1 (0.34) KDM4EGAAALDH1A1NPSR1HPGD
SCHEMBL2548493 0.73 MEN1 (0.44) KDM4EGAAALDH1A1NPSR1HPGD
SCHEMBL8767378 0.73 CYP11B1 (0.48) GAAMEN1MAPTGABRA1CNR1
SCHEMBL7194022 0.72 PTGDR2 (0.43) CYP19A1KDM4EGAAALDH1A1NPSR1
SCHEMBL2722893 0.72 TRPV4 (0.52) KDM4EGAAALDH1A1NPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440643-B1 FLUORINATED 4''-CYANO SUBSTITUTED TERPHENYLS SECR DEFENCE BRIT (GB) 1997-09-03 EP claimed