SCHEMBL8769683

SCHEMBL8769683

CCCOc1ccc(CCC(=O)N2CCOCC2)cc1C1=Nc2c(c(C)nn2CCC)C(=O)[N]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.39
NPC1 O15118 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
GLA P06280 1/20 0.39
FKBP1A P62942 3/20 0.38
PDE5A O76074 1/20 0.36
TSHR P16473 2/20 0.36
TP53 P04637 2/20 0.35
LMNA P02545 1/20 0.35
ALDH1A1 P00352 4/20 0.34
TLR8 Q9NR97 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
HTT P42858 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 4/20 0.34
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7795495 0.83 NPC1 (0.48) RAB9ANPC1KDM4EHPGDPDE5A
SCHEMBL3841327 0.77 PDE5A (0.59) PDE5A
SCHEMBL6930144 0.69 RAB9A (0.38) RAB9ANPC1KDM4EHPGDGLA
SCHEMBL6933205 0.68 RAB9A (0.39) RAB9ANPC1KDM4EHPGDGLA
SCHEMBL6933209 0.63 PKM (0.41) RAB9ANPC1KDM4EHPGDGLA
SCHEMBL6638843 0.62 PDE5A (0.54) PDE5ALMNAALDH1A1HTTKMT2A
SCHEMBL9097067 0.61 PDE5A (0.47) PDE5A
SCHEMBL10195739 0.60 FKBP1A (0.72) RAB9AFKBP1ATSHRTP53ALDH1A1
SCHEMBL9426298 0.60 FKBP1A (0.53) RAB9ANPC1KDM4EHPGDGLA
SCHEMBL8984884 0.59 LMNA (0.63) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793498-A1 BICYCLIC HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF IMPOTENCE Pfizer Limited (GB) 1997-09-10 EP claimed
WO-1996016657-A1 BICYCLIC HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF IMPOTENCE PFIZER LIMITED (GB) 1996-06-06 WO claimed
EP-0793498-A1 BICYCLIC HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF IMPOTENCE Pfizer Limited (GB) 1997-09-10 EP disclosed
WO-1996016657-A1 BICYCLIC HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF IMPOTENCE PFIZER LIMITED (GB) 1996-06-06 WO disclosed