SCHEMBL8769884

SCHEMBL8769884

O=C1NC(=O)C(C[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)N1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.57
IDO1 P14902 2/20 0.51
TDO2 P48775 1/20 0.51
CTSL P07711 13/20 0.49
CTSK P43235 12/20 0.49
CTSS P25774 8/20 0.48
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
TACR1 P25103 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29080074 0.76 IDO1 (0.64) IDO1TDO2
SCHEMBL13964643 0.75 IDO1 (0.51) IDO1TDO2CTSLCTSKCTSS
SCHEMBL6093916 0.75 CTRB1 (0.72) CTRB1CTSLCTSKCTSSTACR1
SCHEMBL6093920 0.75 CTRB1 (0.72) CTRB1CTSLCTSKCTSSTACR1
SCHEMBL2482903 0.75 CTRB1 (0.76) CTRB1CTSLCTSKCTSSTACR1
SCHEMBL2435512 0.75 CTRB1 (0.76) CTRB1CTSLCTSKCTSSTACR1
SCHEMBL1051352 0.75 CTRB1 (0.76) CTRB1CTSLCTSKCTSSTACR1
SCHEMBL8766141 0.74 IDO1 (0.57) IDO1TDO2
SCHEMBL8900969 0.73 CTRB1 (0.74) CTRB1CTSLCTSKCTSSTACR1
SCHEMBL18320645 0.73 CTRB1 (0.74) CTRB1CTSLCTSKCTSSTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793673-A1 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR Takeda Chemical Industries, Ltd. (JP) 1997-09-10 EP disclosed
WO-1996016079-A2 ALPHA-KETOAMIDE DERIVATIVES AS CATHEPSIN L INHIBITOR TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1996-05-30 WO disclosed