SCHEMBL8771793

SCHEMBL8771793

CC1=C(c2ccccc2)c2cc(C(=O)O)ccc2C(C)(C)C1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RARB P10826 15/20 0.48
RARG P13631 14/20 0.48
RARA P10276 13/20 0.48
RXRA P19793 5/20 0.47
NR2E1 Q9Y466 1/20 0.46
PDK2 Q15119 1/20 0.41
KMO O15229 1/20 0.41
CYP26A1 O43174 1/20 0.40
CYP26B1 Q9NR63 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8771941 0.87 RARA (0.66) RARBRARGRARACYP26A1CYP26B1
SCHEMBL12365183 0.76 SRD5A2 (0.53) KMO
SCHEMBL485022 0.75 TDP2 (0.50) RARBRARGRARARXRACYP26A1
SCHEMBL8771650 0.74 RARB (0.77) RARBRARGRARARXRANR2E1
SCHEMBL8028154 0.72 RXRA (0.59) RARBRARGRARARXRACYP26A1
SCHEMBL8771833 0.70 RARB (0.52) RARBRARGRARARXRANR2E1
SCHEMBL8771825 0.69 RARB (0.41) RARBRARGRARARXRANR2E1
SCHEMBL17275573 0.69 RARB (0.50) RARBRARGRARARXRANR2E1
SCHEMBL8028156 0.68 RARA (0.60) RARBRARGRARARXRANR2E1
SCHEMBL2744011 0.68 GRIK1 (0.57) RARBRARGRARARXRAKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661259-B1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL MYERS SQUIBB CO (US) 1997-10-08 EP disclosed
US-5648385-A TREATING RHEUMATOID ARTHRITIS BRISTOL-MYERS SQUIBB CO. (US) 1997-07-15 US disclosed
US-5618839-A Retinoid-like compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-08 US disclosed
EP-0661259-A1 Substituted (5,6)-dihydronaphthalenyl compounds having retinoid-like activity BRISTOL-MYERS SQUIBB COMPANY (US) 1995-07-05 EP disclosed