SCHEMBL8772402

SCHEMBL8772402

O=C1CC([S+]([O-])Cc2ccccc2)N1CCCCCCc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
SLC6A3 Q01959 1/20 0.39
CHRM1 P11229 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
MCOLN3 Q8TDD5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8439618 0.93 GSK3A (0.43) CYP1A2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8772475 0.92 FAAH (0.42) CYP1A2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8553197 0.91 HTR2A (0.40) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8772398 0.89 GSK3A (0.39) CYP1A2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8772495 0.88 GSK3A (0.41) HTR2AMEN1KMT2AGSK3AGSK3B
SCHEMBL8772498 0.87 HTT (0.39) MEN1KMT2AALDH1A1GAA
SCHEMBL8619484 0.87 GSK3B (0.39) CYP1A2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8443653 0.83 KMT2A (0.46) KDM4EMEN1KMT2AALDH1A1
SCHEMBL8772523 0.83 HCRTR1 (0.43) MEN1KMT2AGSK3AGSK3BALDH1A1
SCHEMBL8555803 0.83 HRH3 (0.41) DRD2DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799200-A1 SUBSTITUTED AZETIDIN-2-ONES FOR TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-10-08 EP disclosed