SCHEMBL8772717

SCHEMBL8772717

B.N#Cc1ccc(OCC2(O)CN3CCC2CC3)cc1

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.43
HRH3 Q9Y5N1 8/20 0.41
HRH2 P25021 5/20 0.41
HRH1 P35367 5/20 0.41
MMP13 P45452 5/20 0.41
TRPM8 Q7Z2W7 1/20 0.39
TRPV4 Q9HBA0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8772629 0.97 SIGMAR1 (0.43) SIGMAR1HRH3HRH2HRH1MMP13
SCHEMBL8417820 0.87 FDFT1 (0.37) MMP13
SCHEMBL8968385 0.85 MMP13 (0.39) MMP13
Hydrochloric Acid SCHEMBL8418615 0.84 FDFT1 (0.37) MMP13
Hydrochloric Acid SCHEMBL8968667 0.75 LTA4H (0.42) HRH3MMP13
Hydrochloric Acid SCHEMBL8422025 0.75 LTA4H (0.44) HRH3
SCHEMBL8594298 0.74 CHRM2 (0.48)
SCHEMBL8969436 0.70 MMP13 (0.38) MMP13
SCHEMBL227294 0.69 HRH3 (0.45) SIGMAR1HRH3HRH2HRH1TRPM8
SCHEMBL14292185 0.67 KMT2A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691349-A ANTICHOLESTEROL AGENTS; ATHEROSCLEROSIS ZENECA LIMITED (GB) 1997-11-25 US disclosed
EP-0654032-B1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LTD (GB) 1997-10-15 EP disclosed
EP-0654032-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS. ZENECA LTD (GB) 1995-05-24 EP disclosed
WO-1994003451-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1994-02-17 WO disclosed