SCHEMBL8774435

SCHEMBL8774435

CCCOc1ccc(C#Cc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACACB O00763 18/20 0.40
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA7 P36544 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774463 0.96 MCHR1 (0.41) ACACBHSD17B10
SCHEMBL8774602 0.94 ACACB (0.39) ACACBLMNAHTTCHRNB2CHRNB4
SCHEMBL8774095 0.92 NR5A1 (0.41) ACACBLMNAHTT
SCHEMBL8775170 0.91 CYP2D6 (0.46) LMNAHTTHSD17B10
SCHEMBL8774805 0.89 NQO1 (0.41) ACACB
SCHEMBL8775031 0.85 CYP11B1 (0.39) ACACBLMNAHSD17B10CHRNA7
SCHEMBL8774387 0.82 APP (0.46) ACACB
SCHEMBL9154867 0.82 ACACB (0.41) ACACBLMNAHTTHSD17B10CHRNB2
SCHEMBL8774528 0.80 ACACB (0.42) ACACBHTTCHRNB2CHRNB4CHRNA3
SCHEMBL8774295 0.80 FFAR1 (0.44) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed