SCHEMBL8774387

SCHEMBL8774387

COc1ccc(C#Cc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.46
KCNH2 Q12809 1/20 0.41
TRPV3 Q8NET8 1/20 0.39
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
BACE1 P56817 1/20 0.37
ACACB O00763 2/20 0.35
MCHR1 Q99705 1/20 0.35
PDE4D Q08499 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
HAO1 Q9UJM8 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774805 0.85 NQO1 (0.41) CYP11B1CYP11B2ACACB
SCHEMBL8774435 0.82 ACACB (0.40) ACACB
SCHEMBL8774602 0.82 ACACB (0.39) APPACACBL3MBTL1ALDH1A1
SCHEMBL8775031 0.81 CYP11B1 (0.39) CYP11B1CYP11B2ACACBMCHR1ALDH1A1
SCHEMBL8774095 0.80 NR5A1 (0.41) ACACBL3MBTL1ALDH1A1
SCHEMBL9159082 0.79 APP (0.47) APPKCNH2TRPV3CYP11B1CYP11B2
SCHEMBL8775170 0.79 CYP2D6 (0.46) MCHR1L3MBTL1ALDH1A1
SCHEMBL8774463 0.79 MCHR1 (0.41) ACACBMCHR1ALDH1A1
SCHEMBL8774297 0.78 FFAR1 (0.40) ACACB
SCHEMBL19999378 0.76 APP (0.47) APPKCNH2ACACBMCHR1PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed