SCHEMBL8774805

SCHEMBL8774805

CCOc1ccc(C#Cc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.41
ACACB O00763 15/20 0.38
SYK P43405 1/20 0.38
FFAR1 O14842 1/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8775031 0.96 CYP11B1 (0.39) NQO1ACACBSYKFFAR1CYP11B1
SCHEMBL8774602 0.89 ACACB (0.39) ACACB
SCHEMBL8774435 0.89 ACACB (0.40) ACACB
SCHEMBL8774095 0.86 NR5A1 (0.41) ACACBTSHR
SCHEMBL8774463 0.85 MCHR1 (0.41) ACACB
SCHEMBL8775170 0.85 CYP2D6 (0.46)
SCHEMBL8774387 0.85 APP (0.46) ACACBCYP11B1CYP11B2
SCHEMBL8774297 0.82 FFAR1 (0.40) ACACBFFAR1
SCHEMBL9159722 0.81 NQO1 (0.42) NQO1ACACBTSHRTDP1
SCHEMBL8774295 0.79 FFAR1 (0.44) ACACBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed