SCHEMBL8774602

SCHEMBL8774602

CCCCOc1ccc(C#Cc2cc(F)c(F)nc2F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.39
CYP2D6 P10635 3/20 0.39
CYP3A4 P08684 1/20 0.39
CYP19A1 P11511 4/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C9 P11712 3/20 0.38
CYP2C19 P33261 3/20 0.38
LTA4H P09960 3/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA7 P36544 1/20 0.37
CHRNA4 P43681 1/20 0.37
APP P05067 1/20 0.36
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
NR5A1 Q13285 1/20 0.36
HPGD P15428 3/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774095 0.97 NR5A1 (0.41) ACACBCYP2D6CYP3A4CYP19A1CYP1A2
SCHEMBL8775170 0.96 CYP2D6 (0.46) CYP2D6CYP3A4CYP19A1CYP1A2CYP2C9
SCHEMBL8774435 0.94 ACACB (0.40) ACACBCHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL8774463 0.91 MCHR1 (0.41) ACACBCYP2D6CYP3A4CYP1A2HPGD
SCHEMBL8774805 0.89 NQO1 (0.41) ACACB
SCHEMBL8775031 0.85 CYP11B1 (0.39) ACACBCHRNA7HPGDLMNARAB9A
SCHEMBL8774821 0.83 FFAR1 (0.43) RARARARBRAB9ASMN1; SMN2
SCHEMBL8774387 0.82 APP (0.46) ACACBAPPALDH1A1L3MBTL1
SCHEMBL8774374 0.82 FFAR1 (0.42) CYP3A4RARARARBLMNAKDM4E
SCHEMBL9158222 0.82 ACACB (0.40) ACACBCYP2D6CYP3A4CYP19A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed