SCHEMBL8774513

SCHEMBL8774513

CCc1ccc(-c2ccc(CCc3cc(F)c(F)nc3F)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.39
CYP17A1 P05093 1/20 0.36
CYP21A2 P08686 1/20 0.36
CYP11B1 P15538 1/20 0.36
GPR84 Q9NQS5 1/20 0.35
MAOB P27338 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
RARB P10826 2/20 0.34
RARA P10276 1/20 0.34
RARG P13631 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
FAAH O00519 1/20 0.32
GCGR P47871 1/20 0.32
MAPK14 Q16539 1/20 0.32
DHFR P00374 1/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
TP53 P04637 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8775165 0.95 TAAR1 (0.42) TAAR1GPR84L3MBTL1DHFRNPC1
SCHEMBL8774334 0.91 NPC1 (0.40) TAAR1CYP17A1CYP21A2CYP11B1MAOB
SCHEMBL8774250 0.88 RARB (0.44) RARBRARARARGSMN1; SMN2NPC1
SCHEMBL8774036 0.87 RARB (0.49) RARBRARARARGSMN1; SMN2MAPK14
SCHEMBL8774829 0.85 RAB9A (0.36) GPR84SMN1; SMN2NPC1GAARAB9A
SCHEMBL8774157 0.84 RAB9A (0.39) GPR84L3MBTL1SMN1; SMN2DHFRNPC1
SCHEMBL8774498 0.83 HTR2A (0.40) GPR84RARBRARARARGSMN1; SMN2
SCHEMBL8774847 0.82 ACACB (0.43) L3MBTL1RARBRARASMN1; SMN2DHFR
SCHEMBL8774925 0.82 CYP2D6 (0.46) L3MBTL1RARBRARASMN1; SMN2NPC1
SCHEMBL8774823 0.81 HTR2A (0.46) RARBRARARARGMAPK14TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed