SCHEMBL8774157

SCHEMBL8774157

CCOc1ccc(-c2ccc(CCc3cc(F)c(F)nc3F)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.39
MAPT P10636 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NQO1 P15559 1/20 0.38
KDM4E B2RXH2 4/20 0.38
NPC1 O15118 3/20 0.38
LMNA P02545 2/20 0.38
FFAR1 O14842 2/20 0.38
ALDH1A1 P00352 2/20 0.38
GPR84 Q9NQS5 1/20 0.38
PPARD Q03181 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
FFAR4 Q5NUL3 2/20 0.37
DHFR P00374 1/20 0.37
CDC25A P30304 1/20 0.37
CDC25B P30305 1/20 0.37
CDC25C P30307 1/20 0.37
DUSP3 P51452 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
HSD17B10 Q99714 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774796 0.96 NQO1 (0.41) NQO1KDM4ELMNAALDH1A1GPR84
SCHEMBL8774925 0.90 CYP2D6 (0.46) RAB9AMAPTL3MBTL1KDM4ENPC1
SCHEMBL8774847 0.90 ACACB (0.43) RAB9AMAPTL3MBTL1KDM4ENPC1
SCHEMBL8774330 0.87 CYP3A4 (0.43) RAB9AMAPTL3MBTL1LMNAALDH1A1
SCHEMBL8775001 0.85 PKM (0.42) LMNAALDH1A1SMN1; SMN2CHRNA7
SCHEMBL8774833 0.85 LMNA (0.44) RAB9AMAPTL3MBTL1NPC1LMNA
SCHEMBL8774513 0.84 TAAR1 (0.39) RAB9AL3MBTL1NPC1LMNAGPR84
SCHEMBL8774334 0.84 NPC1 (0.40) RAB9AMAPTNPC1SMN1; SMN2HSD17B10
SCHEMBL8774813 0.83 MEN1 (0.42) LMNAALDH1A1SMN1; SMN2
SCHEMBL9155765 0.82 RAB9A (0.40) RAB9AMAPTL3MBTL1NQO1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed