SCHEMBL8774556

SCHEMBL8774556

CCc1ccc(C#Cc2cnc(Cl)c(Cl)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 5/20 0.47
TDP1 Q9NUW8 2/20 0.42
CYP2A6 P11509 1/20 0.39
FFAR1 O14842 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ACACB O00763 1/20 0.36
ALDH1A1 P00352 3/20 0.36
NPSR1 Q6W5P4 2/20 0.36
RET P07949 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774695 0.88 FFAR1 (0.43) EGLN1TDP1FFAR1ACACBALDH1A1
SCHEMBL8774593 0.85 FFAR1 (0.41) EGLN1TDP1FFAR1L3MBTL1ACACB
SCHEMBL8774237 0.84 HSD17B10 (0.42) FFAR1L3MBTL1ALDH1A1LMNA
SCHEMBL8774402 0.83 ALDH1A1 (0.51) ACACBALDH1A1LMNAPOLB
SCHEMBL8774497 0.80 ACACB (0.43) L3MBTL1ACACBALDH1A1NPSR1LMNA
SCHEMBL8774397 0.80 NPC1 (0.47) L3MBTL1ACACBALDH1A1LMNAPOLB
SCHEMBL9158538 0.78 FFAR1 (0.59) EGLN1TDP1CYP2A6FFAR1L3MBTL1
SCHEMBL8774773 0.78 ALDH1A1 (0.50) L3MBTL1ACACBALDH1A1LMNAPOLB
SCHEMBL8774742 0.77 CHRNB2 (0.36) EGLN1TDP1FFAR1ACACB
SCHEMBL8774736 0.77 CHRNB2 (0.36) EGLN1TDP1FFAR1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed