SCHEMBL8774007

SCHEMBL8774007

CCCc1ccc(-c2cc(F)c(F)nc2Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
TP53 P04637 1/20 0.42
PKM P14618 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPT P10636 1/20 0.37
GFER P55789 1/20 0.37
RARB P10826 3/20 0.36
ALDH1A1 P00352 1/20 0.36
NISCH Q9Y2I1 1/20 0.35
MAOB P27338 2/20 0.34
CNR2 P34972 2/20 0.34
CNR1 P21554 1/20 0.34
ALOX5 P09917 1/20 0.34
CTRC Q99895 1/20 0.34
PTGS2 P35354 1/20 0.34
MCL1 Q07820 1/20 0.33
RARA P10276 1/20 0.33
RARG P13631 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774419 0.91 RARB (0.43) RAB9ANPC1TP53SMN1; SMN2MAPT
SCHEMBL8775053 0.90 RARB (0.48) RAB9ASMN1; SMN2HSD17B10MAPTRARB
SCHEMBL8774679 0.89 RARB (0.50) RAB9ATP53SMN1; SMN2HSD17B10MAPT
SCHEMBL8774744 0.88 GCGR (0.38) RAB9ANPC1TP53PKMSMN1; SMN2
SCHEMBL8774599 0.86 NPC1 (0.41) RAB9ANPC1TP53PKMSMN1; SMN2
SCHEMBL8774928 0.84 NPC1 (0.40) RAB9ANPC1TP53PKMSMN1; SMN2
SCHEMBL8775158 0.83 GPR84 (0.34) RAB9ANPC1TP53PKMSMN1; SMN2
SCHEMBL8775154 0.83 GPR84 (0.34) RAB9ANPC1TP53PKMSMN1; SMN2
SCHEMBL8775089 0.81 GPR84 (0.36) MAPTRARBMAOBCTRCRARA
SCHEMBL8775095 0.81 GPR84 (0.36) MAPTRARBMAOBCTRCRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed