SCHEMBL8774995

SCHEMBL8774995

CCCCc1ccc(-c2ccc(-c3cnc(Cl)c(Cl)c3)cc2F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.46
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
NPC1 O15118 4/20 0.41
NFKB1 P19838 3/20 0.41
NFKB2 Q00653 3/20 0.41
RELA Q04206 3/20 0.41
MAPK1 P28482 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
RARA P10276 1/20 0.41
RARG P13631 1/20 0.41
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
CTRC Q99895 1/20 0.39
MAPT P10636 2/20 0.39
S1PR1 P21453 2/20 0.38
S1PR3 Q99500 2/20 0.38
HSD11B1 P28845 1/20 0.36
BRS3 P32247 1/20 0.36
HSD17B10 Q99714 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8774917 0.96 RARB (0.51) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774251 0.95 RARB (0.53) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774831 0.95 RARB (0.53) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL8774671 0.93 NPC1 (0.42) RARBRAB9ASMN1; SMN2NPC1RARA
SCHEMBL8775178 0.87 FEN1 (0.38) GRM2
SCHEMBL8774724 0.86 AKR1C2 (0.50) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL9155955 0.85 RARB (0.48) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL9879667 0.83 RARB (0.46) RARBRAB9ASMN1; SMN2NPC1NFKB1
SCHEMBL19253582 0.82 RARB (0.56) RARBRARARARGAKR1C2AKR1C1
SCHEMBL19253584 0.82 RARB (0.56) RARBRARARARGAKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519370-B1 Heterocyclic derivatives MERCK PATENT GMBH (DE) 1997-11-05 EP disclosed
EP-0519370-A2 Heterocyclic derivatives MERCK PATENT GmbH (DE) 1992-12-23 EP disclosed