SCHEMBL877631

SCHEMBL877631

CN(C(=O)c1ccc2c(c1)C(N1C=CC=C(C(=O)O)C1C(F)(F)F)CC2)C1CCN(c2ccnc(C3CC3)n2)CC1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
HRH4 Q9H3N8 2/20 0.32
HRH3 Q9Y5N1 2/20 0.32
POLB P06746 1/20 0.32
PDK2 Q15119 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878097 0.90 KDM4A (0.35) KDM4AKDM4CHRH4HRH3POLB
SCHEMBL877666 0.90 KDM4A (0.34) KDM4AKDM4CHRH4HRH3POLB
SCHEMBL878580 0.85 ALDH1A1 (0.34) KDM4AKDM4CPDK2
SCHEMBL877844 0.85 F10 (0.37) KDM4AKDM4CPOLBPDK2
SCHEMBL877632 0.77 HRH4 (0.31) KDM4AKDM4CHRH4HRH3POLB
SCHEMBL785366 0.74 WDR5 (0.38)
SCHEMBL876176 0.74 F10 (0.32) PDK2
SCHEMBL877421 0.73 CCR5 (0.36) KDM4AKDM4CPOLB
SCHEMBL785126 0.73 POLB (0.37) POLB
SCHEMBL785562 0.71 ALDH1A1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP claimed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO claimed
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed