SCHEMBL8779180

SCHEMBL8779180

CCCCOc1ccnc(OC(=O)NC(=O)[C@@H](N)Cc2ccccc2)c1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.38
ALOX5 P09917 1/20 0.38
PPARG P37231 1/20 0.38
GALR1 P47211 1/20 0.37
OPRK1 P41145 1/20 0.37
POLB P06746 1/20 0.37
TSHR P16473 1/20 0.37
FAAH O00519 1/20 0.37
AGER Q15109 1/20 0.37
REN P00797 1/20 0.36
CTSK P43235 3/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSH P09668 1/20 0.36
LTA4H P09960 1/20 0.36
CIT O14578 1/20 0.36
CTSC P53634 1/20 0.36
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
ALPI P09923 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779203 0.97 OPRK1 (0.37) OPRK1FAAHCTSKCTSLCTSB
SCHEMBL8779263 0.97 OPRK1 (0.37) OPRK1FAAHCTSKCTSLCTSB
SCHEMBL8779075 0.95 OPRK1 (0.41) PPARGOPRK1CITCTSCOPRM1
SCHEMBL8779351 0.91 OPRK1 (0.40) OPRK1POLBCITCTSCOPRM1
SCHEMBL8779204 0.87 KDM4E (0.39) OPRK1LTA4HCITCTSCOPRD1
SCHEMBL8779164 0.87 KDM4E (0.39) OPRK1LTA4HCITCTSCOPRD1
SCHEMBL8779188 0.86 CTSC (0.37) OPRK1CITCTSCOPRM1OPRD1
SCHEMBL8779157 0.85 XIAP (0.40) FAAHXIAP
SCHEMBL8885111 0.85 POLB (0.40) GALR1OPRK1POLBTSHRAGER
SCHEMBL8779165 0.82 XIAP (0.38) OPRK1RENXIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed