SCHEMBL8779203

SCHEMBL8779203

CCCCCOc1ccnc(OC(=O)NC(=O)[C@H](N)Cc2ccccc2)c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 2/20 0.37
MEN1 O00255 1/20 0.37
NR1I2 O75469 1/20 0.37
LMNA P02545 1/20 0.37
CHRM2 P08172 1/20 0.37
CYP3A4 P08684 1/20 0.37
ADRA2A P08913 1/20 0.37
MAPT P10636 1/20 0.37
HTR2B P41595 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KMT2A Q03164 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CNR2 P34972 1/20 0.36
TYR P14679 2/20 0.36
CTSK P43235 3/20 0.36
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSH P09668 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779263 1.00 OPRK1 (0.37) OPRK1MEN1NR1I2LMNACHRM2
SCHEMBL8779180 0.97 PTGES (0.38) OPRK1CTSKCTSLCTSBCTSH
SCHEMBL8779075 0.94 OPRK1 (0.41) OPRK1CYP3A4MAPTCITCTSC
SCHEMBL8779351 0.90 OPRK1 (0.40) OPRK1CITCTSCOPRM1OPRD1
SCHEMBL8779204 0.86 KDM4E (0.39) OPRK1CYP3A4CITLTA4HCTSC
SCHEMBL8779164 0.86 KDM4E (0.39) OPRK1CYP3A4CITLTA4HCTSC
SCHEMBL8779165 0.86 XIAP (0.38) OPRK1MEN1NR1I2LMNACHRM2
SCHEMBL8882433 0.85 PTPN1 (0.42) OPRK1MEN1NR1I2LMNACHRM2
SCHEMBL8779188 0.85 CTSC (0.37) OPRK1CYP3A4CITCTSCOPRM1
SCHEMBL8779157 0.82 XIAP (0.40) LMNACYP3A4S1PR1S1PR3FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed