SCHEMBL8779075

SCHEMBL8779075

CCCOc1ccnc(OC(=O)NC(=O)[C@@H](N)Cc2ccccc2)c1O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 2/20 0.41
PPARG P37231 6/20 0.40
MAPT P10636 1/20 0.37
CTSC P53634 1/20 0.37
CIT O14578 1/20 0.37
ALPI P09923 1/20 0.36
PKM P14618 1/20 0.36
PTGS1 P23219 1/20 0.36
XIAP P98170 1/20 0.36
SLC7A5 Q01650 1/20 0.36
AKT1 P31749 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
GPR142 Q7Z601 2/20 0.36
SLC15A1 P46059 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779180 0.95 PTGES (0.38) OPRK1PPARGCTSCCITALPI
SCHEMBL8779263 0.94 OPRK1 (0.37) OPRK1MAPTCTSCCITCYP3A4
SCHEMBL8779203 0.94 OPRK1 (0.37) OPRK1MAPTCTSCCITCYP3A4
SCHEMBL8779351 0.92 OPRK1 (0.40) OPRK1CTSCCITALPIPKM
SCHEMBL8779164 0.88 KDM4E (0.39) OPRK1CTSCCITALPIPKM
SCHEMBL8779204 0.88 KDM4E (0.39) OPRK1CTSCCITALPIPKM
SCHEMBL8779188 0.87 CTSC (0.37) OPRK1CTSCCITALPIPKM
SCHEMBL8779136 0.85 IKBKB (0.37) PPARGMAPTXIAPALDH1A1SLC15A1
SCHEMBL8885435 0.84 OPRK1 (0.43) OPRK1PPARGMAPTCTSCCIT
SCHEMBL8779198 0.80 LTA4H (0.46) MAPTXIAPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed