SCHEMBL8779351

SCHEMBL8779351

CCOc1ccnc(OC(=O)NC(=O)[C@@H](N)Cc2ccccc2)c1O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 5/20 0.40
OPRM1 P35372 3/20 0.40
OPRD1 P41143 3/20 0.40
PKM P14618 2/20 0.38
ALPI P09923 1/20 0.38
PTGS1 P23219 1/20 0.38
XIAP P98170 1/20 0.38
SLC7A5 Q01650 1/20 0.38
CTSC P53634 1/20 0.38
CIT O14578 1/20 0.38
AKT1 P31749 1/20 0.37
SLC15A1 P46059 1/20 0.37
GPR142 Q7Z601 2/20 0.37
POLB P06746 1/20 0.37
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2C Q14957 1/20 0.36
MMP8 P22894 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8779075 0.92 OPRK1 (0.41) OPRK1OPRM1OPRD1PKMALPI
SCHEMBL8779180 0.91 PTGES (0.38) OPRK1OPRM1OPRD1PKMALPI
SCHEMBL8779203 0.90 OPRK1 (0.37) OPRK1OPRM1OPRD1CTSCCIT
SCHEMBL8779263 0.90 OPRK1 (0.37) OPRK1OPRM1OPRD1CTSCCIT
SCHEMBL8779204 0.90 KDM4E (0.39) OPRK1OPRD1PKMALPIPTGS1
SCHEMBL8779164 0.90 KDM4E (0.39) OPRK1OPRD1PKMALPIPTGS1
SCHEMBL8779188 0.88 CTSC (0.37) OPRK1OPRM1OPRD1PKMALPI
SCHEMBL8779212 0.84 HPGD (0.38) POLBGRIN3BGRIN1GRIN2C
SCHEMBL8779176 0.84 HPGD (0.38) POLBGRIN3BGRIN1GRIN2C
SCHEMBL8881760 0.84 OPRK1 (0.43) OPRK1OPRM1OPRD1PKMALPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661269-B1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AG (DE) 1997-03-26 EP disclosed
EP-0661269-A1 Substituted heterocyclic carboxylic acid amides, their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-07-05 EP disclosed